DYRK

Inhibitory Selectivity

Isoform-specific Inhibitors

DYRK Products

New DYRK Products
Catalog No. Information Product Use Citations Product Validations
S7338

AZ191

AZ191 is a potent and selective DYRK1B inhibitor with IC50 of 17 nM in a cell-free assay, about 5- and 110-fold selectivity over DYRK1A and DYRK2, respectively.

S7327

ID-8

ID-8 is a DYRK inhibitor, and sustains embryonic stem cell self-renewal in long-term culture.

S3406New

LDN-192960

LDN-192960 (Compd 1) is a potent inhibitor of Haspin and Dual-specificity Tyrosine-regulated Kinase 2 (DYRK2) with IC50 of 10 nM and 48 nM, respectively.

Catalog No. Information Product Use Citations Product Validations
S7338

AZ191

AZ191 is a potent and selective DYRK1B inhibitor with IC50 of 17 nM in a cell-free assay, about 5- and 110-fold selectivity over DYRK1A and DYRK2, respectively.

S7327

ID-8

ID-8 is a DYRK inhibitor, and sustains embryonic stem cell self-renewal in long-term culture.

S3406New

LDN-192960

LDN-192960 (Compd 1) is a potent inhibitor of Haspin and Dual-specificity Tyrosine-regulated Kinase 2 (DYRK2) with IC50 of 10 nM and 48 nM, respectively.