Endothelin Receptor

Inhibitory Selectivity

Isoform-specific Inhibitors

Endothelin Receptor Products

Catalog No. Information Product Use Citations Product Validations
S0017

Lu-135252

Lu-135252 (Darusentan,HMR-4005) is a selective endothelin A receptor (ET-A receptor) antagonist indicated for the oral treatment of resistant hypertension.

S6665

Sparsentan (PS-433540, RE-021)

Sparsentan (PS-433540, RE-021, DARA) is a dual endothelin type A receptor(ETA) and angiotensin II type 1 receptor antagonist.

Catalog No. Information Product Use Citations Product Validations
S0017

Lu-135252

Lu-135252 (Darusentan,HMR-4005) is a selective endothelin A receptor (ET-A receptor) antagonist indicated for the oral treatment of resistant hypertension.

S6665

Sparsentan (PS-433540, RE-021)

Sparsentan (PS-433540, RE-021, DARA) is a dual endothelin type A receptor(ETA) and angiotensin II type 1 receptor antagonist.