LTR
Inhibitory Selectivity
Isoform-specific Inhibitors
LTR Products
| Catalog No. | Information | Product Use Citations | Product Validations |
|---|---|---|---|
| S8126 |
MK571MK571 (L660711) is a selective, orally active CysLT1 receptor(Cysteinyl leukotriene receptor) antagonist. |
HepG2 cells were exposed to ETV (5 μM and 20 μM) alone or in combination with the efflux transporter inhibitors LY335979 (P-gp, 5 μM), KO143 (BCRP, 5 μM), and MK571 (MRP, 10 μM).
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| S2959New |
LY255283LY255283 is an antagonist of leukotriene B4 (LTB4) receptor (BLT2) that displaces [3H]LTB4 from its binding site on lung membranes with pKi of 7.0. |
| Catalog No. | Information | Product Use Citations | Product Validations |
|---|---|---|---|
| S8126 |
MK571MK571 (L660711) is a selective, orally active CysLT1 receptor(Cysteinyl leukotriene receptor) antagonist. |
HepG2 cells were exposed to ETV (5 μM and 20 μM) alone or in combination with the efflux transporter inhibitors LY335979 (P-gp, 5 μM), KO143 (BCRP, 5 μM), and MK571 (MRP, 10 μM).
|
|
| S2959New |
LY255283LY255283 is an antagonist of leukotriene B4 (LTB4) receptor (BLT2) that displaces [3H]LTB4 from its binding site on lung membranes with pKi of 7.0. |
