OX Receptor

Inhibitory Selectivity

Isoform-specific Inhibitors

OX Receptor Products

New OX Receptor Products
Catalog No. Information Product Use Citations Product Validations
S1545

SB408124

SB408124 is a non-peptide antagonist for OX1 receptor with Ki of 57 nM and 27 nM in both whole cell and membrane, respectively, exhibits 50-fold selectivity over OX2 receptor.

S6726New

MK1064

MK1064 is a selective orexin 2 receptor antagonist (2-SORA) with an IC50 of 18 nM.

Catalog No. Information Product Use Citations Product Validations
S1545

SB408124

SB408124 is a non-peptide antagonist for OX1 receptor with Ki of 57 nM and 27 nM in both whole cell and membrane, respectively, exhibits 50-fold selectivity over OX2 receptor.

S6726New

MK1064

MK1064 is a selective orexin 2 receptor antagonist (2-SORA) with an IC50 of 18 nM.