PAR

Inhibitory Selectivity

Isoform-specific Inhibitors

PAR Products

New PAR Products
Catalog No. Information Product Use Citations Product Validations
S9915New

FSLLRY-NH2 TFA

FSLLRY-NH2 TFA (FSY-NH2) is a selective protease-activated receptor 2 (PAR2) inhibitor with an ic50 of 50 µM in PAR2-KNRK cells.

S2916

ML161 (Parmodulin 2)

ML161 (Parmodulin 2) is an allosteric inhibitor of PAR1 with IC50 of 0.26 μM.

S9744New

AZ3451

AZ3451 is a potent antagonist of protease-activated receptor 2 (PAR2) that binds to a remote allosteric site outside the helical bundle with IC50 of 23 nM.

Catalog No. Information Product Use Citations Product Validations
S9915New

FSLLRY-NH2 TFA

FSLLRY-NH2 TFA (FSY-NH2) is a selective protease-activated receptor 2 (PAR2) inhibitor with an ic50 of 50 µM in PAR2-KNRK cells.

S2916

ML161 (Parmodulin 2)

ML161 (Parmodulin 2) is an allosteric inhibitor of PAR1 with IC50 of 0.26 μM.

Catalog No. Information Product Use Citations Product Validations
S9744New

AZ3451

AZ3451 is a potent antagonist of protease-activated receptor 2 (PAR2) that binds to a remote allosteric site outside the helical bundle with IC50 of 23 nM.