ETK/BMX
Inhibitory Selectivity
ETK/BMX Products
Catalog No. | Information | Product Use Citations | Product Validations |
---|---|---|---|
S8422New |
BMX-IN-1BMX-IN-1 is a selective, irreversible inhibitor of bone marrow tyrosine kinase on chromosome X (BMX) targeting cysteine 496 (Cys496) located at the ATP-binding site, with an IC50 of 138 nM for wild-type BMX, also potently inhibits the related Bruton’s tyrosine kinase (BTK) with an IC50 of 10.4 nM. |
Catalog No. | Information | Product Use Citations | Product Validations |
---|---|---|---|
S8422New |
BMX-IN-1BMX-IN-1 is a selective, irreversible inhibitor of bone marrow tyrosine kinase on chromosome X (BMX) targeting cysteine 496 (Cys496) located at the ATP-binding site, with an IC50 of 138 nM for wild-type BMX, also potently inhibits the related Bruton’s tyrosine kinase (BTK) with an IC50 of 10.4 nM. |