Melanocortin Receptor

Inhibitory Selectivity

Melanocortin Receptor Products

New Melanocortin Receptor Products
Catalog No. Information Product Use Citations Product Validations
P1108New

Bremelanotide Acetate

Bremelanotide Acetate (PT-141 Acetate) is a melanocortin receptor (MCR) agonist recently approved in the USA for the treatment of premenopausal women with acquired, generalized hypoactive sexual desire disorder (HSDD), as characterized by low sexual desire that causes marked distress or interpersonal difficulty.

S0019

JNJ-10229570

JNJ-10229570 (UNII-N9IX402L35) is a potent MC1R and MC5R antagonist.

E1002New

Setmelanotide (RM-493)

Setmelanotide (RM-493, BIM-22493, CAM 4072) is a cyclic peptide full agonist of melanocortin-4 receptor (MC4R) with an EC50 of 0.27 nM and a Ki of 2.1 nM.

Catalog No. Information Product Use Citations Product Validations
P1108New

Bremelanotide Acetate

Bremelanotide Acetate (PT-141 Acetate) is a melanocortin receptor (MCR) agonist recently approved in the USA for the treatment of premenopausal women with acquired, generalized hypoactive sexual desire disorder (HSDD), as characterized by low sexual desire that causes marked distress or interpersonal difficulty.

Catalog No. Information Product Use Citations Product Validations
S0019

JNJ-10229570

JNJ-10229570 (UNII-N9IX402L35) is a potent MC1R and MC5R antagonist.

Catalog No. Information Product Use Citations Product Validations
E1002New

Setmelanotide (RM-493)

Setmelanotide (RM-493, BIM-22493, CAM 4072) is a cyclic peptide full agonist of melanocortin-4 receptor (MC4R) with an EC50 of 0.27 nM and a Ki of 2.1 nM.