Neurokinin Receptor

Inhibitory Selectivity

Isoform-specific Inhibitors

Neurokinin Receptor Products

Catalog No. Information Product Use Citations Product Validations
S0772

L-732138

L-732138 (L-732,138) is a selective, potent and competitive antagonist of neurokinin-1 (NK-1) receptor/substance P (SP) receptor. L-732138 inhibits the binding of 125I-SP to the human NK-1 receptor stably expressed in CHO cells with IC50 of 2.3 nM.

Catalog No. Information Product Use Citations Product Validations
S0772

L-732138

L-732138 (L-732,138) is a selective, potent and competitive antagonist of neurokinin-1 (NK-1) receptor/substance P (SP) receptor. L-732138 inhibits the binding of 125I-SP to the human NK-1 receptor stably expressed in CHO cells with IC50 of 2.3 nM.